4.

A. Lang, Naturwissenschaften 43, 257, 284
(1956).
7. S. P. Johnson, W. C. Hall, J. L. Liverman,

8.
9.

unpublished experiments.

, Phystol. Plantarum 9, 389 (1956).
The gibbereilins used were kindly supplied by
the following: Reed A. Gray, division of microbiological research, Merck and Co., Rahway, N.J.; Frank H. Stodola, Northern Uctilization Research Branch, U.S. Department of
Agriculture, Peoria, Il.; and P. C. Marth,
Horticultural Crops Research Branch, U.S.
Department of Agriculture, Beltsville, Md.
10. This investigation was supported in part by
grant No. G-1165 from the National Science
Foundation to J, L. Liverman.
14 February 1957

direct effects of itodoacctate and iodoacetamide on the aerobic oxidation of

pyruvate and cycle intermediates ‘by
mitochondria would provide more information on their effects on respiration
and give a basis for the judicious use of
a particular concentration of these inhibitors to inhibit specifically the glycolytic pathway.

ric measurement of oxygen uptake were

distinct inhibition with all substrates,

the strongest inhibition being observed
in the oxidation of pyruvate and a-keto-

«Iodoacetate and iodoacetamide have

glutarate, which may indicate the sensitivity of systems involving coenzyme A
and lipoic acid. However, the lower con-

the site of inhibition being at the triosephosphate dehydrogenase. Early reports

bitions which cannot be ignored in respiratory studies. It may be noted that
iodoacctate was generally more effective

been used as specific inhibitors of the
Embden-Meyerhof pathwayof glycolysis,
(1) indicated that iodoacetate at low

concentrations inhibited anaerobic glycolysis and respiration with glucose but
not the oxygen uptake induced by addition of pyruvate or lactate. More recent

studies (2) have shown that the oxidation of pyruvate may be reasonably sensitive to iodoacetate. A study of the

Table 1. Effects of iodoacetate and iodoacetamide on the mitochondrial oxidation
of various substrates. The reaction medium

contained 121 mM KCl, 20 mM potas-

sium phosphate buffer (#H 6.8), 0.01 mf
cytochrome c, 5 mAf MgCh, 1mM adenosine monophosphate, 0.5 mM adenosine
triphosphate, and 5 mM substrate. The
temperature was 37°C, The mitochondrial
suspension was incubated for 10 minutes
with the inhibitors in the medium, and
the oxygen uptake was determined over

a period of 1 hour.

centrations also produced definite inhi-

than iodoacetamide. In order to produce

complete inhibition of triose-phosphate
dehydrogenase and glycolysis, concentrations of 0.2 to 0.5 mdf must be used ‘in

most cases, and thus the present results
indicate that a complete inhibition of

glycolysis is usually accompanied with

some effect on respiration (4).
Wintiam C. YANG
Department of Pharmacology,
School of Medicine, University of
Southern California, Los Angeles
References and Notes
1. H. A. Krebs, Brockem. Z. 234. 278 (1931); O.
Meyerhof and E. Boyland, ibid. 237, 406 (1931).
2, P. J. Heald, Biochem. jf, (London) 55, 625
(1953); J. L. Webb, P. R. Saunders, C. H.
Thienes, Arch, Biochem. and Biophys., 22, 458
(1949); G. G. Laties, ibid. 20, 284 (1949).
3. C. M. Montgomery and J. L. Webb, J. Biol.
Chem. 221, 359 (1956).
4. This work was supported by the Life Insurance
Medical Research Fund and aided by facilities
supplied by the Allan Hancock Foundation.
18 February 1957

Change (%) at various
0.01
mAL

0.10
mM

Todoacetate

a-Ketoglutarate
Malate
Pyruvate +
malate
Succinate
Citrate
Isocitrate

—- 6.3

-33.3

-— 75.6

- 4.3
- 38
+ 46
415.0

-43.0
- 8.0
- 81
-15.3

— 85.6
-61.2
-34.6
—35.0

-

7.4

—20.0

Todoacetamide

a-Ketoglutarate
Malate
Pyruvate +
malate
Succinate
Citrate
Isocitrate

31 MAY 1957

1.0
mM

~- 63.9

- 64

-17.2

— 76.3

- 94
- 25
-16.1

-12.6
-17.0
-14.9

—79.7
-—43.1
-—44.1

-

£0

-12.0

-21.0

-.7,3

-35.3

-29.1

Carompound bon

:

(Coune’mun

(atom/

suet

mole) Found TheLactose

12

Maltol

6

Formic acid
Furfuryl

alcohol
©
Naphthyl

i

Lac-

tose/
prod-

8.7

353

14

cn

ory

ratio

104

1/0.51

17.4

5

O82

20.9

urethane
16
3,9-Dinitrobenzoate
12

0.0

6.5

0.0

8.7

1/0.81

1/0.04+

* Based on molar transfer of 1 atom of C44,

atoms 2 through 6 in the glucose moiety
of lactose

(3). Maltol results rather

uniquely from the heat-induced interac-

tion of reducing disaccharides with amino
compounds (2). It has been detected in
evaporated milk, baked cereals, bread
crust, and roasted malt, among other
places (4).

The three compoundsin question were

recovered and purified from heated
(121°C for 4 hours) condensed skim
milk (30 percent total solids) to which
lactose-1-C14
(National
Bureau
of
Standards) had been added. Steam distillation was used to isolate the com-

pounds from the heated milk. Maltol
and furfuryl alcohol were recovered from
this distillate by ethyl ether extraction
and were purified as described clsewhcre
(3, 5). Formic acid was recovered by

neutralizing a portion of the distillate to
pH 7.5 and evaporating the solution to

dryness under vacuum (6). The crude
formate wasselectively converted to CO,
by the method of Osburn e¢ al. (7). This
CO,, samples of furfuryl alcohol and its
derivatives, maltol and lactose, the latter

from the unheated product, were con-

concentrations

Substrate

C

chondrial suspension and the manomet-

summarized in Table |. Both inhibitors
at a concentration of 1.0 mM produced

Uptake of Heart Mitochondria

Activity of BaCos

The preparation of the rat heart mito-

made according to the methods of Montgomery and Webb (3). The results are

Effect of Iodoacetate and
Todoacetamide on Oxygen

Table 1. Levels of C™ activity found
some heat-degradation products of ski
milk containinglastose-1-C™.

Carbon-14 Activity of Some

Heat-Degradation Products of
Milk Containing Lactose-1-C!*
The course of heat-induced lactoseprotein interaction in milk has been followed with the aid of lactose-1-C1* (7).

Use of labeled lactose also appeared at-

tractive for investigation of the sugar’s
decomposition under these conditions.
Of the many fragments known to be
formed (2), formic acid, furfuryl alcohol, and maltol (3-hydroxy-2-methylpyronc-4) were evaluated in these experiments. It has been proposed that
formic acid is derived from carbon atom
No. ! and furfurvl alcohol from carbon

verted to BaCO, (8). Radioactivity in
these preparations was determined with

a windowless flow gas Geiger-Miiller
counter and decade scaling unit.
The data thus secured (Table 1} re-

veal that carbon atom No. | of lactose is
involved in the formic acid and maltol,
but not in the furfuryl alcohol. A preliminary experiment yielded essentially
the same findings with the exception that
some activity was detected in the furfuryl
alcohol (9). Further investigation of the
alcohol and two carefully authenticated
derivatives of it, as shown in Table |,
revealed that it had no activity.
Under the rigorous heating conditions
emploved in these experiments, a number of carbon sources could contribute to
formate; however, carbon 1 of lactose
1087

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